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PRESTO-Tango GPCRome screening (NMUR1)
Assay data:1 Tested
SummaryRelated BioAssays by Target
Agonist activity at human NMUR1 expressed in CHO cells at 1000 nM by calcium mobilization assay relative to control
SummaryPubMed CitationRelated BioAssays by Target
Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Partial agonist activity at human NMUR1 expressed in CHO cells assessed as intrinsic activity at 10^-6 to 10^-12 M by calcium mobilization assay relative to control
Agonist activity at human NMUR1 expressed in CHO cells assessed as intrinsic activity at 10^-6 to 10^-12 M by calcium mobilization assay relative to control
Assay data:2 Tested
Agonist activity at human NMUR1 expressed in CHO cells at 10 nM by calcium mobilization assay relative to control
Assay data:3 Tested
Agonist activity at human NMUR1 expressed in CHO cells at 100 nM by calcium mobilization assay relative to control
Agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Agonist activity at human NMUR1 expressed in CHO cells at 10 nM by calcium mobilization assay
Agonist activity at human NMUR1 expressed in CHO cells at 100 nM by Fluo-4-AM dye based calcium mobilization assay
Assay data:1 Active, 3 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Agonist activity at human NMUR1 expressed in CHO cells at 1 nM by Fluo-4-AM dye based calcium mobilization assay
Agonist activity at human NMUR1 expressed in CHO cells at 10 nM by Fluo-4-AM dye based calcium mobilization assay
Assay data:5 Tested
Activity at human NMU1 receptor up to 10 uM
Activity at human NMU1 receptor at 10 uM
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Agonist activity at human NMUR1 expressed in CHO cells assessed as increase in intracellular calcium influx after 180 secs by Fluo 4-AM dye based FLIPR assay
Assay data:15 Active, 1 Activity ≤ 1 nM, 20 Activity ≤ 1 µM, 20 Tested
Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux after 18 hrs by Fluo-4 AM dye based FLIPR assay
Assay data:2 Active, 2 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux at 100 nM after 18 hrs by Fluo-4 AM dye based FLIPR assay relative to NMU
Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux at 0.1 nM after 18 hrs by Fluo-4 AM dye based FLIPR assay relative to NMU
Assay data:4 Active, 4 Tested
Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux at 0.1 to 10 nM after 18 hrs by Fluo-4 AM dye based FLIPR assay relative to NMU
Assay data:6 Active, 6 Tested
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