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Cross screening panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of OATP1B1 (unknown origin) upto 10000 nM
SummaryPubMed CitationRelated BioAssays by Target
Substrate activity at human OATP1B1 in CHO cells using 14C-labeled ligand
Inhibition of human OATP1B1
Substrate activity at OATP1B1 (unknown origin)
Inhibition of OATP1B1 (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Assay data:6 Active, 2 Activity ≤ 1 µM, 9 Tested
Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for 30 mins followed by [3H]-pitavastatin addition and measured after 2 mins by liquid scintillation analysis
Assay data:4 Active, 2 Activity ≤ 1 µM, 5 Tested
In Vitro Uptake Transporter Assay from US Patent US9090657: "Compound and methods for its production"
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Assay data:7 Active, 6 Activity ≤ 1 µM, 8 Tested
Inhibition of OATP1B1 (unknown origin) at 500 nM
Assay data:7 Tested
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells
Inhibition of human OATP1B1-mediated [3H]-Estrone sulfate uptake expressed in human HepG2 cells at 2 uM
Assay data:6 Tested
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