Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Panlabs assay PDE10A2
Assay data:1 Tested
SummaryRelated BioAssays by Target
3H-cAMP and 3H-cGMP Scintillation Proximity Assay (PDE10A)
Inhibition of full-length recombinant human PDE10A by scintillation proximity assay
Assay data:6 Active, 4 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 6 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of PDE10A2 (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of human recombinant PDE10A expressed in Sf9 cells incubated for 60 mins by scintillation counter analysis
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of PDE10A (unknown origin) by scintillation proximity assay
Inhibition of PDE10A (unknown origin)
Assay data:18 Active, 5 Activity ≤ 1 nM, 18 Activity ≤ 1 µM, 18 Tested
Inhibition of human PDE10A (449 to 789 residues) expressed in Escherichia coli BL21(DE3) using cAMP as substrate at 4 uM incubated for 30 mins by HTRF analysis relative to control
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of human PDE10A (449 to 789 residues) expressed in Escherichia coli BL21(DE3) using cAMP as substrate incubated for 30 mins by HTRF analysis
Binding affinity to PDE10A (unknown origin) assessed as dissociation constant
Assay data:2 Active, 2 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
Binding affinity to full length human PDE10A assessed as dissociation constant
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to full length human PDE10A assessed as dissociation constant using [3H]-cAMP as substrate
Assay data:9 Active, 5 Activity ≤ 1 nM, 9 Activity ≤ 1 µM, 9 Tested
Inhibition of human PDE10A
Assay data:2 Active, 3 Activity ≤ 1 µM, 3 Tested
Inhibition of human PDE10
Inhibition of human recombinant PDE10A using [3H]-cAMP as substrate incubated for 30 mins by radiometric based liquid scintillation analysis
Inhibition of PDE10A (unknown origin) at 1 uM relative to control
Assay data:2 Tested
Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on