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EPHB3 SGC Tm panel (DSF)
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000736a EPHB3
Selectivity interaction (KinomeScan (Eurofins)) EUB0000250b EPHB3
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000143b EPHB3
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Kinobeads competition assays (Proteomics)) EUB0000143b EPHB3
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Thermal Shift Assay. Domain: start/stop: D616-S910
Assay data:27 Tested
Inhibition of human wild type partial length EPHB3 (Q599 to T928 residues) expressed in bacterial expression system assessed as remaining activity at 1 uM relative to control
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of full length Nano-luc fused EPHB3 in human HEK-293T cells incubated for 2 hrs by cell based NanoBRET target engagement assay
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
EPHB3 DiscoveRx kinase panel
EphB3(h) Kinase panel
Inhibition of EPHB3 (unknown origin) at 1 uM
Kinase Assay from Article 10.1021/cb300729y: "De novo design of protein kinase inhibitors by in silico identification of hinge region-binding fragments."
Assay data:2 Active, 6 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
KinomeScan assay: inhibition of EPHB3
Assay data:1 Active, 108 Tested
EphB3(EPB3LGRJ) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
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