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Selectivity interaction (KinomeScan (DiscoverX)) EUB0000702a GRK4
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of human wild type full length GPRK4 (M1 to C578 residues) expressed in bacterial expression system assessed as remaining activity at 1 uM relative to control
SummaryPubMed CitationRelated BioAssays by Target
GRK4 DiscoveRx kinase panel
Inhibition of GRK4 (unknown origin) at 1 uM
KinomeScan assay: inhibition of GRK4
Assay data:1 Active, 108 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
GRK4(GRK4LGRI) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
GRK4 ProQinase selectivity panel
GRK4 Kinase screen
GRK4 Invitrogen selectivity data (BI)
GRK4 SelectScreen Kinase panel (LifeTechnologies)
GRK4 Invitrogen kinase panel
GRK4 Invitrogen Lab (UK) kinase screen (BI)
Inhibition of wild-type human full length GRK4 (M1 to C578 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control
Inhibition of human GRK4 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assay
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of GRK4 (unknown origin) assessed as residual activity measured at 1 uM
Assay data:3 Tested
Inhibition of human GRK4 assessed as percent of control at 2000 nM by KINOMEscan assay relative to control
Inhibition of DNA-tagged human GRK4 assessed as percent of control at 50000 nM by qPCR analysis relative to control
Inhibition of human GRK4 assessed as percent of control at 1000 nM by KINOMEscan assay relative to control
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