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Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as decrease in Vmax using glucose as substrate by Lineweaver-Burk double reciprocal plot analysis
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as decrease in Vmax using ATP as substrate by Lineweaver-Burk double reciprocal plot analysis
Binding affinity to recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as dissociation constant measured after 15 mins by microscale thermophoresis assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Km using 12.5 uM glucose as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.64 mM)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Km using 6.25 uM glucose as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.64 mM)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Km using 3.125 uM glucose as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.64 mM)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Vmax using 12.5 uM glucose as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.012 OD/min)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Vmax using 6.25 uM glucose as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.012 OD/min)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Vmax using 3.125 uM glucose as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.012 OD/min)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Km using 12.5 uM ATP as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 1.62 mM)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Km using 6.25 uM ATP as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 1.62 mM)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Km using 3.125 uM ATP as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 1.62 mM)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Vmax using 12.5 uM ATP as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.019 OD/min)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Vmax using 6.25 uM ATP as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.019 OD/min)
Non competitive inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) assessed as Vmax using 3.125 uM ATP as substrate by Lineweaver-Burk double reciprocal plot analysis (Rvb = 0.019 OD/min)
Inhibition of recombinant human HK2 expressed in Escherichia coli BL21(DE3) using glucose as substrate preincubated for 10 mins followed by substrate addition in presence of ATP by G6PDH/NADP coupled assay
Assay data:2 Active, 21 Tested
Competitive-inhibition of HK2 (unknown origin) assessed as Km at 10 uM using varying levels of glucose-6-phosphate dehydrogenase as substrate by Lineweaver-burk plot analysis
Assay data:3 Tested
Inhibition of HK2 (unknown origin) using glucose-6-phosphate dehydrogenase as substrate preincubated for 10 mins followed by substrate addition
Assay data:2 Active, 4 Tested
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Inhibition of recombinant human HK2 using [U-14C]-labeled glucose as substrate in presence of ATP and NADP by G6PD enzyme coupled spectrophotometric assay
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