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Covalent binding affinity to estrogen receptor alpha assessed as change in molecular weight after 30 mins by electrospray ionization mass spectrometry
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Antagonist activity at estrogen receptor alpha expressed in human HEC1 cells assessed as inhibition of 100 nM estradiol-induced transcriptional activity after 24 hrs by luciferase reporter gene assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Displacement of [3H]estradiol from human estrogen receptor alpha/estrogen receptor beta
Displacement of [3H]estradiol from human estrogen receptor alpha/estrogen receptor beta relative to estradiol
Inhibition of estradiol-induced coactivator peptide SRC1 binding to estrogen receptor alpha expressed in human HEC1 cells at 20 uM after 24 hrs by beta-galactosidase based mammalian two-hybrid assay
Assay data:17 Tested
Antagonist activity at estrogen receptor alpha expressed in human HEC1 cells assessed as inhibition of estradiol-induced transcriptional activity at 20 uM after 24 hrs by beta-galactosidase reporter gene assay
Inhibition of estradiol-induced coactivator peptide SRC1 binding to estrogen receptor alpha expressed in human HEC1 cells after 24 hrs by luciferase based mammalian two-hybrid assay
Assay data:11 Active, 17 Tested
Antagonist activity at estrogen receptor alpha expressed in human HEC1 cells assessed as inhibition of 1 nM estradiol-induced transcriptional activity after 24 hrs by luciferase reporter gene assay
Assay data:14 Active, 1 Activity ≤ 1 µM, 17 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of estradiol-induced coactivator peptide SRC binding to recombinant estrogen receptor by fluorescence polarization assay
Assay data:3 Tested
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