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Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AMC as a substrate measured over 30 mins by Cheng-prusoff equation analysis
Assay data:8 Active, 20 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15 assessed as reduction in free AMC release using Z-FR-AMC as a substrate measured over 30 mins by fluorometric assay
Assay data:7 Active, 20 Tested
Inhibition of Plasmodium falciparum FP-2
Assay data:1 Active, 1 Tested
Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins by fluorimetric assay
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in bacterial expression system using ZFR-AMC as substrate at 100 uM measured for 30 mins by fluorimetric assay relative to control
Assay data:17 Tested
Inhibition of Plasmodium falciparum falcipain-2 preincubated for 30 mins followed by Z-Leu-Arg-AMC substrate addition and measured up to 15 mins by spectrofluorometric analysis
Assay data:11 Active, 11 Tested
Inhibition of Plasmodium falciparum N-terminal His6-tagged falcipain-2 (35 residues) expressed in Escherichia coli M15 pREP4 using Z-Lue-Arg-AMC as substrate measured after 30 mins by spectrofluorometric method
Assay data:16 Active, 14 Activity ≤ 1 µM, 20 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescence assay
Assay data:10 Active, 5 Activity ≤ 1 µM, 17 Tested
Inhibition of Plasmodium falciparum falcipain 2 assessed as second order inactivation rate constant using Z-Phe-Arg-AMC as substrate by fluorometric assay
Assay data:3 Tested
Inhibition of Plasmodium falciparum falcipain 2 at 20 uM using Z-Phe-Arg-AMC as substrate by fluorometric assay relative to control
Assay data:19 Tested
Inhibition of Plasmodium falciparum falcipain 2 using Z-Phe-Arg-AMC as substrate by fluorometric assay
Assay data:3 Active, 2 Activity ≤ 1 µM, 7 Tested
Irreversible inhibition of Plasmodium falciparum falcipain-2 using Cbz-Phe-Arg-AMC as substrate pretreated for 30 mins followed by substrate addition and measured for 30 mins by dialysis method
Assay data:3 Active, 3 Tested
Reversible inhibition of Plasmodium falciparum falcipain-2 using Cbz-Phe-Arg-AMC as substrate pretreated for 30 mins followed by substrate addition and measured for 30 mins by dialysis method
Inhibition of Plasmodium falciparum falcipain-2 assessed as second-order rate constant using Cbz-Phe-Arg-AMC as substrate measured for 15 mins by spectrofluorimetric method
Assay data:20 Tested
Inhibition of Plasmodium falciparum falcipain-2 using Cbz-Phe-Arg-AMC as substrate measured for 15 mins by spectrofluorimetric method
Assay data:4 Active, 3 Activity ≤ 1 µM, 14 Tested
Inhibition of Plasmodium falciparum falcipain-2 at 20 uM using Cbz-Phe-Arg-AMC as substrate measured for 15 mins by spectrofluorimetric method relative to control
Inhibition of Plasmodium falciparum falcipain-2
Assay data:21 Active, 1 Activity ≤ 1 nM, 20 Activity ≤ 1 µM, 29 Tested
Resistance index, ratio of IC50 for falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes to IC50 for falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes
Assay data:16 Tested
Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in bacterial growth after 24 hrs by Giemsa staining based assay
Assay data:4 Active, 1 Activity ≤ 1 µM, 16 Tested
Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction in bacterial growth after 24 hrs by Giemsa staining based assay
Assay data:3 Active, 1 Activity ≤ 1 µM, 16 Tested
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