Related BioAssays, by Target Similarity (List) for PubChem BioAssay (S - PubChem BioAssay - NCBI

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Select item 19635981.

Biochemical Assay from US Patent US20240139197: "INHIBITION OF KDM5A FOR PROMOTING ANTIGEN PRESENTATION, INCREASING CD8+ T CELL INFILTRATION AND BOOSTING ANTI-TUMOR IMMUNE RESPONSE"

Source:: BindingDB

Protein Targets:: Lysine-specific demethylase 4C; ...
Total:: 3

Assay data:13 Active, 13 Activity ≤ 1 µM, 13 Tested

AID:: 1963598

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19340602.

Inhibition of KDM5A (unknown origin ) by TR-FRET assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1934060

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19340573.

Inhibition of Halo-tagged KDM5A PHD3 domain (unknown origin)

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:3 Tested

AID:: 1934057

Summary PubMed Citation Related BioAssays by Target

Select item 19340474.

Inhibition of KDM5A (unknown origin ) demethylase activity using H3 as substrate by Chemiluminescent assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1934047

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19340425.

Inhibition of KDM5A (unknown origin ) by Cellular luciferase reporter assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1934042

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19340416.

Inhibition of KDM5A (unknown origin ) demethylase activity

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested

AID:: 1934041

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19340337.

Inhibition of KDM5A (unknown origin ) by Alphalisa analysis

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:4 Active, 4 Activity ≤ 1 µM, 5 Tested

AID:: 1934033

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19340298.

Inhibition of KDM5A (unknown origin ) by HTMS analysis

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1934029

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19340229.

Inhibition of KDM5A (unknown origin ) by Alphascreen assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:15 Active, 11 Activity ≤ 1 µM, 16 Tested

AID:: 1934022

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 193401810.

Competitive inhibition of KDM5A (unknown origin) in human HeLa cells by TR-FRET assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Tested

AID:: 1934018

Summary PubMed Citation Related BioAssays by Target

Select item 193401611.

Competitive inhibition of KDM5A (unknown origin) in human MM1.S cells by TR-FRET assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Tested

AID:: 1934016

Summary PubMed Citation Related BioAssays by Target

Select item 193401312.

Inhibition of N-terminal his6-tagged human KDM5A (1 to 797 residues) expressed in sf9 insect cells incubated for 20 mins by Alphascreen assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:7 Active, 2 Activity ≤ 1 µM, 8 Tested

AID:: 1934013

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192927313.

Inhibition of KDM5A (unknown origin) using H3K4me3 as substrate by MSD ELISA analysis

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1929273

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191954214.

Biochemical KDM5A Inhibition Assay from US Patent US11691968: "Compound having KDM5 inhibitory activity and pharmaceutical use thereof"

Source:: BindingDB

Protein Targets:: Lysine-specific demethylase 5A; ...
Total:: 1

Assay data:44 Active, 44 Activity ≤ 1 µM, 44 Tested

AID:: 1919542

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 188533015.

Inhibition of KDM5A (unknown origin) in presence of 300 uM 2-OG

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1885330

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 188532916.

Inhibition of KDM5A (unknown origin) in presence of 4 uM 2-OG

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1885329

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 188532417.

Inhibition of recombinant HQ5-Halo-tagged KDM5A PHD3 domain (unknown origin) measured by fluorescence polarization assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:2 Tested

AID:: 1885324

Summary PubMed Citation Related BioAssays by Target

Select item 188531618.

Inhibition of KDM5A (unknown origin) measured by AlphaScreen assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested

AID:: 1885316

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 188528619.

Inhibition of KDM5A (unknown origin) measured by ELISA assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1885286

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 187247020.

Inhibition of full-length KDM5A (1 to 1090 residues)(unknown origin) using ARTK(me3)-QTARKSTGGKAPRKQLA-GGK(biotin) as substrate preincubated for 10 mins followed by substrate addition measured after 45 mins by LANCE Ultra assay

Source:: ChEMBL

Protein Target:: Lysine-specific demethylase 5A

Assay data:1 Active, 1 Tested

AID:: 1872470

Summary Compounds, Active PubMed Citation Related BioAssays by Target

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Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

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