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Inhibition of MEK5 (unknown origin) by discoverX kinomescan assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of MEK5 (unknown origin)
Assay data:3 Tested
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000294b MAP2K5
SummaryRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000714a MAP2K5
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000701a MAP2K5
Selectivity interaction (ScanMAX (DiscoverX)) EUB0000700a MAP2K5
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000305b MAP2K5
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000305b MAP2K5
Selectivity interaction (Enzymatic assay) EUB0000305b MAP2K5
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000321b MAP2K5
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000321b MAP2K5
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000698a MAP2K5
Selectivity interaction (Quantitative chemical proteomics (cell-based phosphorylation and proliferation assays in Hs578t cells)) EUB0000147b MAP2K5
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000147b MAP2K5
Inhibition of MEK5 (unknown origin) expressed in baculovirus expression system incubated for 90 mins in presence of ATP by PKlight ATP detection reagent based luciferase assay
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to wild type human partial length MEK5 (L98 to P448 residues) expressed in mammalian expression system by Kinomescan binding assay
Inhibition of human wild-type partial length MEK5 (L98 to P448 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control
MEK5 DiscoveRx kinase panel
Inhibition of MEK5 (unknown origin) at 1 uM
Inhibition of recombinant human MAP2K5 using Ulight-ARTKQTARKSTGGKAPRKQLAGCG as substrate at 1 uM incubated for 120 mins in presence of ATP by LANCE method relative to control
Assay data:2 Tested
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