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Selectivity interaction (ScanMAX (DiscoverX, competition-binding assay)) EUB0000285b TSSK1B
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (ScanMAX (DiscoverX)) EUB0000285b TSSK1B
Inhibition of STK22D (TSSK1) (unknown origin) at 1 uM relative to control
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of human wild type TSSK1
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of TSSK2 (unknown origin) at 1 uM
TSSK1B DiscoveRx kinase panel
TSSK2(h) Kinase panel
TSSK1(h) Kinase panel
TSSK1(h) Millipore kinase panel
Inhibition of STK22D (unknown origin) at 1 uM
Inhibition of human recombinant TSSK1 assessed as reduction in substrate phosphorylation at 50 to 500 nM using ATP and Ulight-CKKSRGDYMTMQIG (IRS-1) incubated for 60 min by LANCE detection method
Inhibition of TSSK1 (unknown origin) at 3 uM by Z-lyte assay relative to control
Inhibition of TSSK2 (unknown origin) at 3 uM by Z-lyte assay relative to control
Inhibition of TSSK1 (unknown origin) by Z-lyte assay
Inhibition of TSSK2 (unknown origin) by Z-lyte assay
KinomeScan assay: inhibition of TSSK1B
Assay data:108 Tested
TSSK1(TS1BLGP1) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
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