Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
PI3K-gamma Scintillation Proximity Assay from US Patent US11926616: "Aminopyrazine diol compounds as PI3K-γ inhibitors"
Assay data:46 Active, 46 Activity ≤ 1 µM, 46 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Cross screening panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
PIK3CG Invitrogen Lab (UK) kinase screen (BI)
Inhibition of PI3K-gamma (unknown origin) upto 10000 nM
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of recombinant PI5P4Kgamma (unknown origin) expressed in Escherichia coli BL21(DE3) by ADP-Glo reagent based assay
Assay data:42 Tested
Inhibition of PI3Kgamma (unknown origin) using PIP2:PS as substrate preincubated for 1 hr followed by ATP and substate addition and measured after 1 hr by ADP-glo reagent based assay
Assay data:2 Active, 1 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of wild type human PIK3CG in presence of ATP by radiometric kinase assay
Inhibition of wild type human PIK3CG at 1 uM by DiscoverX scanMAX assay relative to control
Antagonist activity at PI3Kgamma (unknown origin) using PIP2 as substrate in presence of ATP incubated for 30 to 60 mins by ADP-glo based luminescence assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Antagonist activity at PI3Kgamma (unknown origin) assessed as inhibition rate at 20 nM using PIP2 as substrate in presence of ATP incubated for 30 to 60 mins by ADP-glo based luminescence assay relative to control
Assay data:29 Tested
Inhibition of PI3Kgamma (unknown origin)
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
Inhibition of P13Kgamma (unknown origin)
Inhibition of PI3Kgamma in mouse RAW264 cells assessed as reduction in LPS-stimulated IL-6 mRNA expression preincubated for 6 hrs followed by LPS addition and measured after 24 hrs by RT-PCR analysis
Inhibition of PI3Kgamma in mouse RAW264 cells assessed as reduction in LPS-stimulated TNFalpha mRNA expression preincubated for 6 hrs followed by LPS addition and measured after 24 hrs by RT-PCR analysis
Inhibition of PI3Kgamma (unknown origin) preincubated for 10 mins followed by ATP addition and measured after 60 mins by ADP-Glo assay
Assay data:1 Active, 3 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of PI3Kgamma (unknown origin) at 10 uM preincubated for 10 mins followed by ATP addition and measured after 60 mins by ADP-Glo assay relative to control
Assay data:3 Tested
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on