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Inhibitory Activity Against KHK In Vitro from US Patent US20240067633: "KETOHEXOKINASE INHIBITOR AND USE THEREOF"
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
KHK-A Assay D from US Patent US11634410: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
KHK-C Assay C from US Patent US11634410: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
Assay data:6 Active, 6 Activity ≤ 1 µM, 6 Tested
KHK-C Assay B from US Patent US11634410: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
KHK-C Assay A from US Patent US11634410: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
Assay data:52 Active, 49 Activity ≤ 1 µM, 53 Tested
Inhibition of KHK (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
KHK Enzyme Activity Assay for Human KHK-C and Human KHK-A from US Patent US11124500: "Disubstituted pyrazole compounds"
Assay data:38 Active, 38 Activity ≤ 1 µM, 38 Tested
Inhibition Assay from US Patent US11083720: "Indazole inhibitors of fructokinase (KHK) and methods of use in treating KHK-mediated disorders or diseases"
Assay data:9 Active, 6 Activity ≤ 1 µM, 9 Tested
Biological Assay from US Patent US10988463: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Assay data:54 Active, 50 Activity ≤ 1 µM, 55 Tested
Biological Assay from US Patent US10787438: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
Assay data:17 Active, 16 Activity ≤ 1 µM, 18 Tested
Enzyme Activity Assay from US Patent US10781212: "2,6-diamino pyridine compounds"
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Enzyme Assay from US Patent US8822447: "Indazole compounds useful as ketohexokinase inhibitors"
Assay data:124 Active, 62 Activity ≤ 1 µM, 154 Tested
Enzyme Assay from US Patent US9771375: "Indazole compounds useful as ketohexokinase inhibitors"
Assay data:126 Active, 64 Activity ≤ 1 µM, 156 Tested
KHK Assay D from US Patent US10174007: "Substituted 3-azabicyclo[3.1.0]hexanes as ketohexokinase inhibitors"
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