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MAP2K1 SGC Tm panel (DSF)
Assay data:1 Tested
SummaryRelated BioAssays by Target
MAP2K2 Invitrogen Lab (UK) kinase screen (BI)
MAP2K1 Invitrogen Lab (UK) kinase screen (BI)
Inhibition of MEK1 (unknown origin) at 1 uM relative to control
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of MEK2 (unknown origin) by discoverX kinomescan assay
Inhibition of MEK1 (unknown origin) by discoverX kinomescan assay
Inhibition of human MEK2
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human MEK1
Inhibition of MAP2K1 (unknown origin) at 1000 nM relative to control
Inhibition of MAP2K1 (unknown origin)
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human full length wild type MEK1 expressed in mammalian system at 1 uM by KINOMEscan analysis relative to control
Inhibition of MEK1 (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Induction of MEK1/2 degradation in human A549 cells assessed as reduction in pERK1/2 levels at 1 to 30 uM incubated for 24 hrs by Western blot analysis
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