Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
BRPF1 SGC Tm panel (DSF)
Assay data:1 Tested
SummaryRelated BioAssays by Target
Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRPF1 (unknown origin) measured after 10 mins by TR-FRET assay
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in bacterial expression system by BROMOscan assay
Assay data:4 Tested
Binding affinity to human partial length BRD1 (E556 to A688 residues) expressed in bacterial expression system by BROMOscan assay
Inhibition of BRPF1 (unknown origin) at 10 uM by DiscoverX BROMOscan assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Displacement of biotinylated JQ1 from BRPF1 bromodomain (unknown origin) incubated for 20 mins by AlphaLISA assay
Binding affinity to BRPF1 bromodomain (unknown origin) incubated for 60 mins by TR-FRET assay
Selectivity interaction (Reader proteins panel (DSF assay)) EUB0000034d BRPF1
Selectivity interaction (Bromodomain panel (DSF assay)) EUB0000323b BRPF1
Selectivity interaction (AlphaScreen) EUB0000323b BRPF1
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Bromodomain panel (DSF assay)) EUB0000323b BRD1
Selectivity interaction (AlphaScreen) EUB0000323b BRD1
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (BROMOscan? panel (DiscoverX)) EUB0000256b BRPF1
Selectivity interaction (BROMOscan? panel (DiscoverX)) EUB0000256b BRD1
Selectivity interaction (TR-FRET assay) EUB0000224e BRPF1
Selectivity interaction (Bromodomain panel (DSF assay)) EUB0000224e BRPF1
Selectivity interaction (AlphaScreen) EUB0000224e BRPF1
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on