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Dopamine D4.2 Eurofins Panlabs panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Binding affinity towards human DRD4 in an in vitro assay with cellular components measured by membrane filtration
Assay data:36 Active, 19 Activity ≤ 1 µM, 233 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]N-methylspiperone from D4 receptor in HEK293 cell membrane assessed as inhibition constant at 10 uM relative to control
Assay data:17 Tested
SummaryPubMed CitationRelated BioAssays by Target
Displacement of [3H]N-methylspiperone from D4 receptor in HEK293 cell membrane
Assay data:51 Active, 1 Activity ≤ 1 nM, 39 Activity ≤ 1 µM, 51 Tested
Partial agonist activity at human D4 receptor expressed in HEK293T cells assessed as inhibition of forskolin-induced cAMP production incubated for 1 hr by HTRF analysis relative to control
Assay data:23 Tested
Partial agonist activity at human D4 receptor expressed in HEK293T cells assessed as inhibition of forskolin-induced cAMP production incubated for 1 hr by HTRF analysis
Assay data:21 Active, 7 Activity ≤ 1 µM, 23 Tested
Partial agonist activity at human D4 receptor assessed as inhibition constant
Assay data:3 Active, 3 Activity ≤ 1 µM, 5 Tested
Agonist activity at D4R (unknown origin)
Agonist activity at D4R (unknown origin) assessed as beta-arrestin recruitment
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Agonist activity at D4R (unknown origin) relative to control
Assay data:3 Tested
Agonist activity at D4R (unknown origin) by camp reporter assay
Assay data:9 Active, 1 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 11 Tested
Displacement of [3H]N-methylspiperone from D4 (unknown origin) receptor expressed in HEK293 cells assessed as inhibition constant
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Displacement of [3H]-methylspiperone from D4 (unknown origin) receptor expressed in HEK293T cells assessed as inhibition constant
Assay data:9 Active, 8 Activity ≤ 1 µM, 9 Tested
Agonist activity at human D4R at 10 uM relative to control
Agonist activity at human D4R
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Displacement of [3H]-spiperone from D4 (unknown origin) receptor expressed in CHO cells assessed as inhibition constant
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to D34 (unknown origin) assessed as inhibition constant
Agonist activity at human D4R expressed in HEK293 cells at 10 uM by calcium flux assay relative to control
Assay data:2 Tested
Agonist activity at human D4R expressed in HEK293 cells by calcium flux assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Displacement of [3H]-spiperone from human D4 receptor assessed as inhibition constant
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