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CK2 Alpha 1 Enzymatic Activity Inhibition from US Patent US11932606: "Anti-cancer/anti-fibrosis compounds"
Assay data:34 Active, 29 Activity ≤ 1 µM, 34 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
CSNK2A2 SGC Tm panel (DSF)
Assay data:1 Tested
SummaryRelated BioAssays by Target
CSNK2A1A SGC Tm panel (DSF)
CSNK2A2A SGC Tm panel (DSF)
CSNK2A1 SGC Tm panel (DSF)
Binding affinity to C-terminal Nano-Luc fused human CK2alpha' expressed in digitonin -permeabilized human HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBRET assay
Assay data:27 Active, 27 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Binding affinity to C-terminal Nano-Luc fused human CK2alpha expressed in digitonin -permeabilized human HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBRET assay
Inhibition of wild type human CK2alpha' in presence of ATP by radiometric kinase assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of wild type human CK2alpha in presence of ATP by radiometric kinase assay
Assay data:1 Active, 2 Tested
Inhibition of wild type human CK2alpha' at 1 uM by DiscoverX scanMAX assay relative to control
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of wild type human CK2alpha at 1 uM by DiscoverX scanMAX assay relative to control
Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBRET assay
Assay data:26 Active, 25 Activity ≤ 1 µM, 27 Tested
Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBRET assay
Assay data:26 Active, 22 Activity ≤ 1 µM, 27 Tested
Inhibition of CK2A2 (unknown origin) by Ambit kinase assay
Assay data:4 Tested
Inhibition of CK2A2 (unknown origin)
Inhibition of CK2A1 (unknown origin)
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