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Inhibition of USP9X (unknown origin) using ubiquitin rhodamine 110 as substrate at 1 to 10 uM by DUBprofiler fluorometric assay
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of human USP9X using ubiquitin rhodamine 110 as substrate at 10 to 50 uM by fluorometric assay
Assay data:1 Tested
Inhibition of human USP9X (1551 to 1970 residues) expressed in Escherichia coli BL21 (DE3) using ubiquitin rhodamine 110 as substrate assessed as remaining enzyme activity at 10 to 50 uM by fluorometric assay
Inhibition of USP9x (unknown origin)
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of USP9X (unknown origin) at 2.5 uM
Inhibition of USP9x (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis
Assay data:6 Tested
Inhibition of USP9X (unknown origin) using Ubiquitin-Rhoadmine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 11 mins by fluorescence assay
Assay data:179 Active, 60 Activity ≤ 1 nM, 160 Activity ≤ 1 µM, 179 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Assay data:58 Active, 38 Activity ≤ 1 nM, 57 Activity ≤ 1 µM, 68 Tested
Inhibition of USP9 (unknown origin) at 10 uM relative to control
Inhibition of USP9 (unknown origin)
Inhibition of human GST-tagged USP9X CD (1554 to 1995 residues) expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine110-glycine using Ubiquitin-Rhodamine110-glycine as substrate by fluorescence based analysis
Inhibition of Usp9x in human MM1S cells at 0.625 to 2.5 uM
SummaryCompounds, ActiveRelated BioAssays by Target
Inhibition of Usp9x in Vemurafenib-resistant human A375R cells assessed as induction of NOXA levels
Inhibition of Usp9x in Vemurafenib-resistant human A375 cells
Inhibition of Usp9x in Vemurafenib-sensitive human A375 cells
Inhibition of Usp9x in primary tumor cells from patient with plasma cell leukemia assessed as reduction in Mcl1 protein levels at 5 uM incubated for 5 to 240 mins relative to control
Inhibition of Usp9x in human MM1.S cells assessed as induction of caspase activity by measuring PARP cleavage at 5 uM incubated for 5 to 240 mins relative to control
Inhibition of Usp9x in human MM1.S cells assessed as reduction in Mcl1 protein levels at 5 uM incubated for 5 to 240 mins relative to control
Inhibition of Usp9x in primary tumor cells from patient with plasma cell leukemia at 5 uM incubated for 60 mins relative to control
SummaryRelated BioAssays by Target
Inhibition of Usp9x in human MM1.S cells at 5 uM incubated for 60 mins relative to control
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