Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
In Vitro Detection of the Inhibitory Activity of Compounds Against PDE 4B Enzyme from US Patent US20240294526: "FUSED TRI-CYCLIC COMPOUND AS A PDE3/PDE4 DUAL INHIBITOR"
Assay data:29 Active, 29 Activity ≤ 1 nM, 29 Activity ≤ 1 µM, 29 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Radioligand Binding Assay from US Patent US12071420: "Pyridine and pyrazine compounds as inhibitors of cannabinoid receptor 2"
Assay data:39 Active, 36 Activity ≤ 1 µM, 39 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Kinase panel (KiNativ target engagement assay in Jurkat cells)) EUB0001635a PRKD2
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (Kinase panel (Z-LYTE Assay)) EUB0001632a PRKD2
Selectivity interaction (Kinase panel (Z-LYTE Assay)) EUB0001632a PRKD1
Selectivity interaction (Kinase panel (Z-LYTE Assay)) EUB0001632a PRKD3
Selectivity interaction (CEREP ligand displacement assays (non-kinase proteins)) EUB0001326b SLC6A4
Selectivity interaction (CEREP ligand displacement assays (non-kinase proteins)) EUB0001326b SLC6A3
Selectivity interaction (CEREP ligand displacement assays (non-kinase proteins)) EUB0001326b SLC6A2
Selectivity interaction (Competition-binding assay (Kinases and other enzymes)) EUB0001326b PRKD3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0001326b PRKD3
Selectivity interaction (Competition-binding assay (Kinases and other enzymes)) EUB0001326b PRKD2
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0001326b PRKD2
Selectivity interaction (KinomeScan (DiscoverX)) EUB0001326b PRKD1
Selectivity interaction (Biochemical dose-response assay (Carna Biosciences)) EUB0001326b PRKD3
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (CARNA Biosciences Kinase Panel (Caliper LabChip3000 mobility shift assay)) EUB0001326b PRKD3
Selectivity interaction (Biochemical dose-response assay (Carna Biosciences)) EUB0001326b PRKD2
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on