BioAssays for PubChem Compound (Select 440317) - PubChem BioAssay - NCBI

Warning: The NCBI web site requires JavaScript to function. more...

Links from PubChem Compound

Items: 16

Select item 16345501.

Inhibition of His6-tagged recombinant human GALK expressed in Escherichia coli HMS174 (DE3) at 5 to 15 uM incubated for 60 mins using galactose and ATP by Kinase-Glo reagent based assay

Source:: ChEMBL

Protein Target:: Galactokinase

Assay data:1 Active, 1 Tested

AID:: 1634550

Summary Compounds, Active Related BioAssays by Target

Select item 13726942.

Agonist activity at human N-terminal HA-tagged P2Y2 receptor expressed in 1321N1 cells

Source:: ChEMBL

Protein Target:: P2Y purinoceptor 2

Assay data:1 Active, 1 Tested

AID:: 1372694

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 9776113.

Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB

Source:: Shanghai Institute of Organic Chemistry

Protein Targets:: Chain 1, Cell division protein ftsZ; ...
Total:: 2972

Assay data:3916 Active, 206 Activity ≤ 1 nM, 1830 Activity ≤ 1 µM, 3916 Tested

AID:: 977611

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Depositor Related BioAssays by Target

Select item 7511934.

Antioxidant activity assessed as inhibiton of Fe2+-induced Fenton reaction-mediated hydroxyl radical formation from H2O2 relative to ATP

Source:: ChEMBL

Assay data:1 Tested

AID:: 751193

Summary PubMed Citation

Select item 7511925.

Antioxidant activity assessed as inhibiton of Fe2+-induced Fenton reaction-mediated hydroxyl radical formation from H2O2 relative to trolox

Source:: ChEMBL

Assay data:1 Tested

AID:: 751192

Summary PubMed Citation

Select item 3029846.

Agonist activity at P2Y11 receptor expressed in 1321N1 cells assessed as cytosolic calcium level

Source:: ChEMBL

Protein Target:: P2Y purinoceptor 11

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 302984

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 1524767.

Antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )

Source:: ChEMBL

Protein Target:: P2X purinoceptor 1

Assay data:11 Active, 6 Activity ≤ 1 µM, 11 Tested

AID:: 152476

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 1504958.

Antagonist activity against phospholipase C coupled rat P2Y purinoceptor 12 (P2Y12)

Source:: ChEMBL

Protein Target:: P2Y purinoceptor 12

Assay data:7 Active, 4 Activity ≤ 1 µM, 12 Tested

AID:: 150495

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 1504899.

Agonist activity against phospholipase C coupled human P2Y purinoceptor 11 (P2Y11)

Source:: ChEMBL

Protein Target:: P2Y purinoceptor 11

Assay data:4 Active, 10 Tested

AID:: 150489

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 15047010.

Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of turkey erythrocytes

Source:: ChEMBL

Protein Target:: P2Y purinoceptor 1

Assay data:14 Active, 1 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 17 Tested

AID:: 150470

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15032111.

Evaluated for agonist activity against phospholipase C coupled recombinant human P2Y purinoceptor 2 (P2Y2)

Source:: ChEMBL

Protein Target:: P2Y purinoceptor 2

Assay data:4 Active, 3 Activity ≤ 1 µM, 12 Tested

AID:: 150321

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15017212.

Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )

Source:: ChEMBL

Protein Target:: P2X purinoceptor 6

Assay data:3 Active, 2 Activity ≤ 1 µM, 7 Tested

AID:: 150172

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15017013.

Antagonist activity against recombinant rat P2X purinoceptor 5 (P2X5)

Source:: ChEMBL

Protein Target:: P2X purinoceptor 5

Assay data:5 Active, 3 Activity ≤ 1 µM, 7 Tested

AID:: 150170

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15016614.

Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 30 uM, expressed in Xenopus oocytes

Source:: ChEMBL

Protein Target:: P2X purinoceptor 4

Assay data:3 Active, 1 Activity ≤ 1 µM, 5 Tested

AID:: 150166

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15015115.

Antagonist activity against recombinant human P2X purinoceptor 3 (P2X3 )

Source:: ChEMBL

Protein Target:: P2X purinoceptor 3

Assay data:9 Active, 1 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 11 Tested

AID:: 150151

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 15014416.

Antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X2) at 10 uM, expressed in Xenopus oocytes

Source:: ChEMBL

Protein Target:: P2X purinoceptor 2

Assay data:4 Active, 1 Activity ≤ 1 µM, 7 Tested

AID:: 150144

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Supplemental Content

Filters: Manage Filters

Refine your results

• What's this?

Target

Proteins (1)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (14)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (3)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (11)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (12)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (15)
BioAssays extracted from the literature
Other (1)
BioAssays deposited by other experimentalists

Actions on your results

View or Download BioAssay in PubChem

Find related data

Recent activity

Clear Turn Off Turn On

BioAssays for PubChem Compound (Select 440317) (16)
PubChem BioAssay

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...

You are here: NCBI > Chemicals & Bioassays > PubChem BioAssay