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Selectivity interaction (GPCR panel (PDSP screen)) EUB0000544a TMEM97
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000544a GABRA1
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000544a SIGMAR1
Selectivity interaction (CSE-HRP surface expression (cell surface expression-horseradish peroxidase assay)) EUB0000544a CFTR
Affinity On-target Cellular interaction (CFTR Restoration Trans-Epithelial Current Clamp (TECC) assay (in HBE cells from F508del CF patients)) EUB0000544a CFTR
Affinity Phenotypic Cellular interaction (Plasma membrane-expressed enzyme acceptor protein (EA-MEM) assay) EUB0000544a CFTR
GPCRScan assay: inhibition of Sigma 2
Assay data:29 Active, 24 Activity ≤ 1 µM, 181 Tested
Corrector activity at HRP-fused CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in matured protein levels at cell surface after 18 to 24 hrs by luminescence assay
Assay data:13 Active, 6 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
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