BioAssays, Active for PubChem Compound (Select 3100) - PubChem BioAssay - NCBI

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Select item 19618571.

Binding affinity towards human CHRM2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M2

Assay data:58 Active, 2 Activity ≤ 1 nM, 37 Activity ≤ 1 µM, 301 Tested

AID:: 1961857

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618562.

Binding affinity towards human DRD3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: D(3) dopamine receptor

Assay data:176 Active, 1 Activity ≤ 1 nM, 87 Activity ≤ 1 µM, 1215 Tested

AID:: 1961856

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618483.

Binding affinity towards human SLC6A2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:123 Active, 40 Activity ≤ 1 µM, 1197 Tested

AID:: 1961848

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618474.

Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:119 Active, 21 Activity ≤ 1 µM, 1213 Tested

AID:: 1961847

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618395.

Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:128 Active, 38 Activity ≤ 1 µM, 927 Tested

AID:: 1961839

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618386.

Binding affinity towards human SLC6A2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:137 Active, 27 Activity ≤ 1 µM, 927 Tested

AID:: 1961838

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19617857.

Compound was evaluated for inhibition of human KCNH2 in an in vitro assay with cellular components measured by membrane filtration, radioactivity method

Source:: ChEMBL

Protein Target:: Potassium voltage-gated channel subfamily H member 2

Assay data:353 Active, 116 Activity ≤ 1 µM, 1804 Tested

AID:: 1961785

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19617838.

Binding affinity towards human HTR6 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 6

Assay data:27 Active, 15 Activity ≤ 1 µM, 148 Tested

AID:: 1961783

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19617829.

Binding affinity towards human HTR5A in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 5A

Assay data:14 Active, 5 Activity ≤ 1 µM, 75 Tested

AID:: 1961782

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196178010.

Binding affinity towards human HTR2C in an in vitro assay with cellular components measured by radioactivity method

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2C

Assay data:123 Active, 1 Activity ≤ 1 nM, 48 Activity ≤ 1 µM, 1199 Tested

AID:: 1961780

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196177911.

Binding affinity towards human HTR2B in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2B

Assay data:103 Active, 70 Activity ≤ 1 µM, 317 Tested

AID:: 1961779

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196177512.

Binding affinity towards human HTR2A in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2A

Assay data:140 Active, 4 Activity ≤ 1 nM, 75 Activity ≤ 1 µM, 414 Tested

AID:: 1961775

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196176813.

Binding affinity towards human HRH2 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: Histamine H2 receptor

Assay data:61 Active, 32 Activity ≤ 1 µM, 283 Tested

AID:: 1961768

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196176614.

Binding affinity towards human HRH1 in an in vitro assay measured by filtration

Source:: ChEMBL

Protein Target:: Histamine H1 receptor

Assay data:151 Active, 1 Activity ≤ 1 nM, 90 Activity ≤ 1 µM, 1239 Tested

AID:: 1961766

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196173915.

Binding affinity towards human DRD3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: D(3) dopamine receptor

Assay data:142 Active, 80 Activity ≤ 1 µM, 896 Tested

AID:: 1961739

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196172616.

Binding affinity towards human CHRM5 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M5

Assay data:19 Active, 13 Activity ≤ 1 µM, 117 Tested

AID:: 1961726

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196172517.

Binding affinity towards human CHRM4 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M4

Assay data:13 Active, 2 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 85 Tested

AID:: 1961725

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196172418.

Binding affinity towards human CHRM3 in an in vitro assay with cellular components measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M3

Assay data:93 Active, 1 Activity ≤ 1 nM, 42 Activity ≤ 1 µM, 1188 Tested

AID:: 1961724

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196172319.

Binding affinity towards human CHRM2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M2

Assay data:155 Active, 74 Activity ≤ 1 µM, 927 Tested

AID:: 1961723

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196172220.

Antagonist activity at human CHRM2 in an in vitro cell-based assay measured by fluorescent imaging plate reader

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M2

Assay data:70 Active, 31 Activity ≤ 1 µM, 1177 Tested

AID:: 1961722

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Target

Proteins (13)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (86)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (31)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (62)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (66)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (3)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Assay Project (7)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (47)
BioAssays extracted from the literature
NIH MLP (11)
BioAssays deposited by the NIH Molecular Libraries Program
Other (27)
BioAssays deposited by other experimentalists

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