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Inhibition of ACK1 (unknown origin)
Assay data:7 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 9 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of NEK11 (unknown origin) assessed as dissociation constant
Assay data:4 Active, 2 Activity ≤ 1 µM, 4 Tested
Inhibition of NEK2 (unknown origin) assessed as dissociation constant
Assay data:8 Active, 5 Activity ≤ 1 µM, 8 Tested
Inhibition of B-Raf V600E mutant (448 to 723 residues) (unknown origin) expressed in Escherichia coli by AlphaScreen assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of B-raf (448 to 723 residues) (unknown origin) expressed in Escherichia coli by AlphaScreen assay
Evaluation of RAF Kinase Activity from US Patent US11492357: "Thieno[3,2-d]pyrimidine derivative compound having inhibitory activity for protein kinase"
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: OCIMY5_PLB cell viability assay
Assay data:980 Active, 10 Activity ≤ 1 nM, 428 Activity ≤ 1 µM, 1912 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Depositor
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: OCIMY7_PLB cell viability assay
Assay data:828 Active, 37 Activity ≤ 1 nM, 590 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: LP1_DSMZ cell viability assay
Assay data:486 Active, 24 Activity ≤ 1 nM, 280 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: MM1S_ATCC cell viability assay
Assay data:1053 Active, 13 Activity ≤ 1 nM, 437 Activity ≤ 1 µM, 1911 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: MMM1_PLB cell viability assay
Assay data:911 Active, 7 Activity ≤ 1 nM, 657 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: KMS12BM_JCRB cell viability assay
Assay data:870 Active, 12 Activity ≤ 1 nM, 424 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: Karpas25_ECACC cell viability assay
Assay data:975 Active, 20 Activity ≤ 1 nM, 350 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: H1112_PLB cell viability assay
Assay data:695 Active, 3 Activity ≤ 1 nM, 231 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: INA6_PLB cell viability assay
Assay data:965 Active, 40 Activity ≤ 1 nM, 443 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: JIM3_ECACC cell viability assay
Assay data:782 Active, 10 Activity ≤ 1 nM, 239 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: KHM11_PLB cell viability assay
Assay data:572 Active, 29 Activity ≤ 1 nM, 524 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: Delta47_JCRB cell viability assay
Assay data:811 Active, 19 Activity ≤ 1 nM, 394 Activity ≤ 1 µM, 1912 Tested
Cytotoxicity against human A-375 cells by MTT assay
Assay data:3 Active, 4 Tested
SummaryCompounds, ActivePubMed Citation
Inhibition of human BRAF V600E mutant using MEK1 as substrate in presence of ATP
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
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