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Human Y1 receptor (Neuropeptide Y receptors)
Assay data:9 Active, 9 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Human NPFF1 receptor (Neuropeptide FF/neuropeptide AF receptors)
Assay data:11 Active, 11 Tested
Human NPFF2 receptor (Neuropeptide FF/neuropeptide AF receptors)
Rat Y1 receptor (Neuropeptide Y receptors)
Assay data:22 Active, 22 Tested
Displacement of (R)-Na-Diphenylacetyl-Nomega[2-([2,3-3H]-propionylamino)ethyl]aminocarbonyl (4-hydroxybenzyl)-argininamide from NPY1R in human SK-N-MC cells
Assay data:3 Active, 2 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]EYF from human NPFF2 expressed in CHO cells by radioligand binding assay
Assay data:2 Active, 1 Activity ≤ 1 µM, 7 Tested
Displacement of [3H]NPVF from human NPFF1 expressed in CHO cells by radioligand binding assay
Assay data:4 Active, 3 Activity ≤ 1 µM, 7 Tested
Displacement of (R)-Na-Diphenylacetyl-Nomega[2-([2,3-3H]-propionylamino)ethyl]aminocarbonyl (4-hydroxybenzyl)-argininamide from NPY1R in human SK-N-MC cells by radioligand binding assay
Assay data:5 Active, 5 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 7 Tested
Displacement of [3H]UR-MK136 from NPY1R in human SK-N-MC cells by radioligand binding assay
Assay data:9 Active, 7 Activity ≤ 1 nM, 9 Activity ≤ 1 µM, 9 Tested
Binding affinity to human NPFF2 receptor expressed in CHO cells
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to human NPFF1 receptor expressed in CHO cells
Antagonist activity at NPY1R in human HEL cells assessed as inhibition of 10 nM pNPY-induced Ca+2 response preincubated for 10 mins by Fura-2 dye based spectrofluorimetric analysis
Assay data:6 Active, 5 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 6 Tested
Antagonist activity at NPY1R in human HEL cells assessed as inhibition of 10 nM pNPY-induced Ca+2 response preincubated for 5 mins by Fura-2 dye based spectrofluorimetric analysis
Antagonist activity at NPY1R in human HEL cells assessed as inhibition of 10 nM pNPY-induced Ca+2 response preincubated for 10 secs by Fura-2 dye based spectrofluorimetric analysis
Assay data:6 Active, 6 Activity ≤ 1 µM, 6 Tested
Displacement of [3H]propionyl-pNPY from NPY1R in HEL cells after 60 to 90 mins by flow cytometric analysis
Assay data:5 Active, 4 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested
Binding affinity to NPY1R in human SK-N-MC cells after 2 hrs by liquid scintillation counting assay
Displacement of [3H]UR-MK114 from human neuropeptide Y receptor type 1 expressed in human SK-N-MC cells
Assay data:30 Active, 28 Activity ≤ 1 µM, 43 Tested
Antagonist activity at neuropeptide Y receptor type 1 in HEL assessed as inhibition of pNPY-induced calcium mobilization by Fura-2 calcium assay
Assay data:10 Active, 2 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 21 Tested
Agonist activity at human NPFF2 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation counting
Assay data:7 Active, 4 Activity ≤ 1 µM, 7 Tested
Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation counting
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
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