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Agonist activity at human ADRB2 in an in vitro cell-based assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:14 Active, 10 Activity ≤ 1 µM, 635 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human liver FBPase expressed in Escherichia coli by spectrophotometry method
Assay data:1 Active, 1 Activity ≤ 1 µM, 3 Tested
Inhibition of recombinant human FBP expressed in expressed Escherichia coli BL21 (DE3) incubated for 1 hr by hanging drop vapour method
Assay data:17 Active, 7 Activity ≤ 1 µM, 17 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Cytotoxicity against paclitaxel-resistant human HCT116tax cells assessed as DNA damage by measuring fluorescence intensity incubated for 30 mins by Hoechst 33342 staining accumulation assay
Assay data:5 Active, 5 Tested
SummaryCompounds, ActivePubMed Citation
Inhibition of recombinant human P-gp ATPase activity in presence of MgATP preincubated for 40 min measured after 20 min by Pgp-Glo assay
Assay data:5 Active, 6 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Cytotoxicity against paclitaxel-resistant human HCT116tax cells assessed as reduction on cell viability at 100 to 200 uM incubated for 48 hrs in presence of paclitaxel by MTT assay
Cytotoxicity against human HCT-116 cells assessed as reduction on cell viability at 100 uM incubated for 48 hrs in presence of paclitaxel by MTT assay
Cytotoxicity against in human HCT-116 cells overexpressing human BCRP assessed as DNA damage by measuring fluorescence intensity at 100 uM incubated for 30 mins by Hoechst 33342 staining accumulation assay
Assay data:6 Active, 6 Tested
Cytotoxicity against human HCT-116 cells overexpressing human MDR1 assessed as DNA damage by measuring fluorescence intensity at 100 uM incubated for 30 mins by Hoechst 33342 staining accumulation assay
Inhibition of human liver FBPase expressed in Escherichia coli BL21(DE3) using FBP as substrate in presence of PGI and G6PDH by spectrophotometric method
Assay data:85 Active, 67 Activity ≤ 1 µM, 91 Tested
Activation of human recombinant AMPK alpha2/beta1/gamma1 using substrate-1 peptide as substrate incubated for 45 mins in presence of ATP by HTRF assay
Assay data:21 Active, 6 Activity ≤ 1 µM, 22 Tested
Inhibition of wild-type full-length human liver FBPase expressed in Escherichia coli BL21 (DE3) using FBP as substrate by malachite green dye based assay
Assay data:30 Active, 8 Activity ≤ 1 µM, 60 Tested
Inhibition of human liver FBP1 incubated for 5 mins by fluorescence method
Assay data:2 Active, 5 Tested
Allosteric activation of AMPK alpha2/beta1/gamma1 in human HepG2 cells by scintillation proximity assay
Assay data:23 Active, 9 Activity ≤ 1 µM, 23 Tested
Inhibition of human FBPase expressed in Escherichia coli BL21 (DE3) using FBP as substrate incubated for 5 mins by malachite green dye based spectrophotometry
Assay data:18 Active, 7 Activity ≤ 1 µM, 19 Tested
ERK5 transcriptional activity HTS
Assay data:60 Active, 2000 Tested
Activation of human recombinant AMPKalpha2beta2gamma2 expressed in Escherichia coli at 10 uM incubated for 1 hr using serine/threonine kinase substrate
Assay data:1 Active, 1 Tested
Activation of human recombinant AMPKalpha2beta2gamma1 expressed in Escherichia coli at 10 uM incubated for 1 hr using serine/threonine kinase substrate
Activation of human recombinant AMPKalpha2beta1gamma3 expressed in Escherichia coli at 10 uM incubated for 1 hr using serine/threonine kinase substrate
Activation of human recombinant AMPKalpha2beta1gamma1 expressed in Escherichia coli at 10 uM incubated for 1 hr using serine/threonine kinase substrate
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