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Binding affinity towards human DRD3 in an in vitro assay with cellular components measured by scintillation counting
Assay data:176 Active, 1 Activity ≤ 1 nM, 87 Activity ≤ 1 µM, 1215 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Compound was evaluated for inhibition of human PTGS2 in an in vitro cell free assay measured by fluorescence spectroscopy
Assay data:79 Active, 12 Activity ≤ 1 µM, 1183 Tested
Binding affinity towards human HTR2C in an in vitro assay with cellular components measured by radioactivity method
Assay data:123 Active, 1 Activity ≤ 1 nM, 48 Activity ≤ 1 µM, 1199 Tested
Antagonist activity at human HTR2A in an in vitro cell-based assay measured by fluorescent imaging plate reader
Assay data:116 Active, 1 Activity ≤ 1 nM, 39 Activity ≤ 1 µM, 1135 Tested
Agonist activity at human HTR1A in an in vitro cell-based assay measured by fluorescent imaging plate reader
Assay data:41 Active, 16 Activity ≤ 1 µM, 1178 Tested
Binding affinity towards human DRD2 in an in vitro assay with cellular components measured by membrane filtration, scintillation proximity assay
Assay data:153 Active, 2 Activity ≤ 1 nM, 73 Activity ≤ 1 µM, 1228 Tested
Agonist activity at human DRD1 in an in vitro cell-based assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:32 Active, 2 Activity ≤ 1 nM, 19 Activity ≤ 1 µM, 1197 Tested
Compound was evaluated for inhibition of human ADRA2C in an in vitro assay with cellular components measured by membrane filtration
Assay data:195 Active, 66 Activity ≤ 1 µM, 1241 Tested
Binding affinity towards human ADRA2B in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:166 Active, 1 Activity ≤ 1 nM, 62 Activity ≤ 1 µM, 1209 Tested
Antagonist activity at human ADRA2A in an in vitro cell-based assay measured by fluorescent imaging plate reader
Assay data:80 Active, 18 Activity ≤ 1 µM, 1172 Tested
Agonist activity at human ADRA1A in an in vitro cell-based assay (NIBR assay) measured by fluorescent imaging plate reader
Assay data:42 Active, 2 Activity ≤ 1 nM, 28 Activity ≤ 1 µM, 969 Tested
Rat 5-HT2A receptor (5-Hydroxytryptamine receptors)
Assay data:45 Active, 45 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Human 5-HT2C receptor (5-Hydroxytryptamine receptors)
Assay data:97 Active, 97 Tested
Rat 5-HT2C receptor (5-Hydroxytryptamine receptors)
Assay data:17 Active, 17 Tested
Human 5-HT2B receptor (5-Hydroxytryptamine receptors)
Assay data:94 Active, 94 Tested
Rat 5-HT1F receptor (5-Hydroxytryptamine receptors)
Assay data:6 Active, 6 Tested
Human 5-HT1F receptor (5-Hydroxytryptamine receptors)
Assay data:40 Active, 40 Tested
Human 5-ht1e receptor (5-Hydroxytryptamine receptors)
Assay data:47 Active, 47 Tested
Human 5-HT1D receptor (5-Hydroxytryptamine receptors)
Assay data:84 Active, 84 Tested
Mouse 5-HT7 receptor (5-Hydroxytryptamine receptors)
Assay data:24 Active, 24 Tested
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