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Inhibition of TGEV 3CL protease using Dabcyl-KTSAVLQ/SGFRKME-Edans as substrate incubated for 30 mins followed by substrate addition measured after 30 mins by FRET assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Antiviral activity against TGEV assessed as log reduction in virus progeny at 4 uM
Assay data:1 Tested
SummaryPubMed Citation
Antiviral activity against TGEV assessed as reduction in virus titre at 4 uM
Inhibition of Transmissible gastroenteritis coronavirus H16 guanine-N7 methyltransferase expressed in Saccharomyces cerevisiae YBS40 (MATa leu2 ade2 trp1 his3 ura3 can1 abd1::hisGp360-ABD1)
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
Antiviral activity against Transmissible gastroenteritis virus infected in pig at 25 mg/animal administered 3 times per day
Antiviral activity against Transmissible gastroenteritis virus infected in ST cells pre-treated 2 hrs before virus infection measured 6 hrs post virus infection by immunofluorescent assay
Assay data:29 Active, 14 Activity ≤ 1 µM, 37 Tested
Antiviral activity against Transmissible gastroenteritis virus infected in ST cells assessed as reduction in N-protein expression pre-treated before virus infection measured 16 hrs post virus infection by Western blotting
Assay data:6 Active, 6 Tested
Antiviral activity against Transmissible gastroenteritis virus infected in ST cells assessed as reduction in caspase-3 activation pre-treated before virus infection measured 16 hrs post virus infection by Western blotting
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as inhibition of S and N protein expression treated 2 hrs before infection measured after 6 hrs post infection by indirect immunofluorescent assay
Assay data:5 Active, 8 Tested
Inhibition of Transmissible gastroenteritis virus TFI recombinant GST-tagged 3C-like protease expressed in Escherichia coli BL21 (DE3)
Assay data:6 Active, 8 Tested
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as protection against virus-induced cytopathic effect at 100 uM after 24 hrs post infection
Assay data:5 Active, 5 Tested
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as protection against virus-induced cytopathic effect at 5 uM after 24 hrs post infection
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as protection against virus-induced cytopathic effect at 100 uM after 18 hrs post infection
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as protection against virus-induced cytopathic effect at 5 uM after 18 hrs post infection
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as protection against virus-induced caspase 3 activation at 5 uM after 18 hrs post infection
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as protection against virus-induced caspase 3 activation at 5 uM after 14 hrs post infection
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as reduction of 3CL protease mRNA level after 6 hrs post infection by RT-PCR
Assay data:2 Tested
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as reduction of N protein mRNA level after 6 hrs post infection by RT-PCR
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as reduction of 3CL protease mRNA level at 10 uM after 6 hrs post infection by RT-PCR
Assay data:3 Tested
Antiviral activity against Transmissible gastroenteritis virus TFI infected in swine testicle cells assessed as reduction of 3CL protease mRNA level at 5 uM after 6 hrs post infection by RT-PCR
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